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FAAH selectively influences placebo effectsPECINA, M; MARTINEZ-JAUAND, M; HODGKINSON, C et al.Molecular psychiatry. 2014, Vol 19, Num 3, pp 385-391, issn 1359-4184, 7 p.Article

Synthesis and biological evaluation of dibenz[b,f][1, 5]oxazocine derivatives for agonist activity at κ-opioid receptorMITRA, Sudipta; TUHIN SUVRO BANERJEE; HOTA, Sandip K et al.European journal of medicinal chemistry. 2011, Vol 46, Num 5, pp 1713-1720, issn 0223-5234, 8 p.Article

Synthesis of 7,9-diazabicyclo[4.2.2]decanes as conformationally restricted K receptor agonists: Fine tuning of the dihedral angle of the ethylenediamine pharmacophoreSUNNAM, Sunil K; RACK, Elisabeth; SCHEPMANN, Dirk et al.European journal of medicinal chemistry. 2011, Vol 46, Num 6, pp 1972-1982, issn 0223-5234, 11 p.Article

The Importance of Alkynyl Chain Presence for the Activity of Adenine Nucleosides/Nucleotides on Purinergic ReceptorsDAL BEN, D; BUCCIONI, M; LAMBERTUCCI, C et al.Current medicinal chemistry. 2011, Vol 18, Num 10, pp 1444-1463, issn 0929-8673, 20 p.Article

The characterization of a novel V1b antagonist lead seriesSMETHURST, Chris A; BORTHWICK, Jennifer A; GAINES, Simon et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 1, pp 92-96, issn 0960-894X, 5 p.Article

hNk2 receptor antagonists. The use of intramolecular hydrogen bonding to increase solubility and membrane permeabilityETTORRE, Alessandro; D'ANDREA, Piero; MAURO, Sandro et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 6, pp 1807-1809, issn 0960-894X, 3 p.Article

Application of Ullmann and Ullmann―Finkelstein reactions for the synthesis of N-aryl-N-(1H-pyrazol-3-yl) acetamide or N-(1-aryl-1H-pyrazol-3-yl) acetamide derivatives and pharmacological evaluationDEPREZ-POULAIN, Rebecca; COUSAERT, Nicolas; TOTO, Patrick et al.European journal of medicinal chemistry. 2011, Vol 46, Num 9, pp 3867-3876, issn 0223-5234, 10 p.Article

Discovery process and pharmacological characterization of a novel dual orexin 1 and orexin 2 receptor antagonist useful for treatment of sleep disordersDI FABIO, Romano; PELLACANI, Annalisa; STASI, Luigi et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 18, pp 5562-5567, issn 0960-894X, 6 p.Article

Identification and optimisation of novel sulfonamide, selective vasopressin V1B receptor antagonistsBAKER, James; BINGHAM, Matilda; NAPIER, Susan et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 12, pp 3603-3607, issn 0960-894X, 5 p.Article

Synthesis and SAR studies of novel 2-(6-aminomethylaryl-2-aryl-4-oxo-quinazolin-3(4H)-yl)acetamide Vasopressin V1b receptor antagonistsNAPIER, Susan E; LETOURNEAU, Jeffrey J; HO, Koc-Kan et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 12, pp 3813-3817, issn 0960-894X, 5 p.Article

Targeting Opioid and Neurokinin-1 Receptors to Treat AlcoholismRODRIGUEZ, F. D; COVENAS, R.Current medicinal chemistry. 2011, Vol 18, Num 28, pp 4321-4334, issn 0929-8673, 14 p.Article

5-OMe-UDP is a Potent and Selective P2Y6-Receptor AgonistGINSBURG-SHMUEL, Tamar; HAAS, Michael; SCHUMANN, Marlen et al.Journal of medicinal chemistry (Print). 2010, Vol 53, Num 4, pp 1673-1685, issn 0022-2623, 13 p.Article

In silico directed chemical probing of the adenosine receptor familyAREIAS, Filipe M; BREA, Jose; GREGORI-PUIGJANE, Elisabet et al.Bioorganic & medicinal chemistry. 2010, Vol 18, Num 9, pp 3043-3052, issn 0968-0896, 10 p.Article

Novel small molecule bradykinin B1 receptor antagonists. Part 3: Hydroxyurea derivativesSCHNATBAUM, Karsten; SCHAUDT, Marco; ZISCHINSKY, Gunther et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 3, pp 1233-1236, issn 0960-894X, 4 p.Article

Probes for narcotic receptor mediated phenomena. 40. N-Substituted cis-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-8-olsIYER, Malliga R; YONG SOK LEE; DESCHAMPS, Jeffrey R et al.Bioorganic & medicinal chemistry. 2010, Vol 18, Num 1, pp 91-99, issn 0968-0896, 9 p.Article

Structure-Based Discovery of Novel Chemotypes for Adenosine A2A Receptor AntagonistsKATRITCH, Vsevolod; JAAKOLA, Veli-Pekka; LANE, J. Robert et al.Journal of medicinal chemistry (Print). 2010, Vol 53, Num 4, pp 1799-1809, issn 0022-2623, 11 p.Article

Subtlety of the Structure-Affinity and Structure—Efficacy Relationships around a Nonpeptide Oxytocin Receptor AgonistFRANTZ, Marie-Céline; RODRIGO, Jordi; BOUDIER, Laure et al.Journal of medicinal chemistry (Print). 2010, Vol 53, Num 4, pp 1546-1562, issn 0022-2623, 17 p.Article

Synthesis and dual PPARα/δ agonist effects of 1,4-disubstituted 1,2,3-triazole analogues of GW 501516CIOCOIU, Calin C; NIKOLIC, Nataša; HUYEN HOA NGUYEN et al.European journal of medicinal chemistry. 2010, Vol 45, Num 7, pp 3047-3055, issn 0223-5234, 9 p.Article

Synthesis and evaluation of opioid receptor-binding affinity of elaeocarpenine and its analogsKURASAKI, Haruaki; OKAMOTO, Iwao; MORITA, Nobuyoshi et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 5, pp 1601-1603, issn 0960-894X, 3 p.Article

Synthesis and theoretical studies on energetics of novel N- and O- perfluoroalkyl triazole tagged thienopyrimidines - Their potential as adenosine receptor ligandsSIRISHA, B; NARSAIAH, B; YAKAIAH, T et al.European journal of medicinal chemistry. 2010, Vol 45, Num 5, pp 1739-1745, issn 0223-5234, 7 p.Article

Synthesis of substituted N-[3-(3-methoxyphenyl)propyl] amides as highly potent MT2-selective melatonin ligandsYUEQING HU; HO, Maurice K. C; CHAN, King H et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 8, pp 2582-2585, issn 0960-894X, 4 p.Article

Tetrahydroindolizinone NK1 antagonistsJIANMING BAO; HUAGANG LU; MILLS, Sander G et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 7, pp 2354-2358, issn 0960-894X, 5 p.Article

Allosteric Enhancers of A1 Adenosine Receptors: State of the Art and New Horizons for Drug DevelopmentROMAGNOLI, R; BARALDI, P. G; TABRIZI, M. A et al.Current medicinal chemistry. 2010, Vol 17, Num 30, pp 3488-3502, issn 0929-8673, 15 p.Article

Discovery and structure-activity relationship of a novel spirocarbamate series of NPY Y5 antagonistsLESLIE, Colin P; BENTLEY, Jonathan; PIZZI, Domenica A et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 20, pp 6103-6107, issn 0960-894X, 5 p.Article

Discovery of 2-aminoimidazopyridine adenosine A2A receptor antagonistsMCGUINNESS, Brian F; COLE, Andrew G; HICKS, Catherine et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 22, pp 6845-6849, issn 0960-894X, 5 p.Article

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